平安! 发表于 2011-11-9 19:57 3 l! T) y0 m6 P, |1 I$ g
Pazopanib (100 mg/kg/day free base equivalent) 7 Y0 j& O4 W& @" L& \" v# |8 a
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
/ g3 J+ ^0 e; B9 [搜索了一下,原料一大堆。7 V! Z! {7 |# C+ p1 s1 |
! i# _* u& }5 j( k& C9 G/ b对不起!100mg/kg是用于移植瘤的,我弄错了。9 W1 W+ A& E" d: b2 _
7 i1 u6 e( G5 V: M: q. a1 [7 ~& d; b7 N以下是正版说明书的推荐用量。 }+ ~- x6 m% f4 ^* W- Y- C! F
t; a/ _2 [$ P3 V--------------------- DOSAGE AND ADMINISTRATION ----------------
+ F, _+ J, i% q1 O% w! g& T7 C* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) % K, d! D4 E1 B$ X
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
" u7 O# \; ^/ A* j---------------------DOSAGE FORMS AND STRENGTHS --------------
5 I* |6 ?, H* t0 z- j( H3 d200 mg tablets. (3)
: C( K' y$ Y8 d1 @: \8 h$ J-------------------------------CONTRAINDICATIONS------------------------ |